human Vasopressin V2 receptor is also validated for Aequorin (calcium), cAMP, radioligand binding competition assays

Target Information

Family :
Vasopressin
Receptor :

V2

Species :
Homo sapiens
Accession number :
NP_000045.1

Assay Information

Cat. Number :
FAST-0552I
Method :
HTRF
Assay Type :
IPOne
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
[Arg8]-Vasopressin
EC50:
6.14nM*
#ALT#

Mode:
antagonist
Reference antagonist:
[Adamantaneacetyl1, O-Et-D-Tyr2, Val4, Aminobutyryl6, Arg8,9]-Vasopressin
IC50:
509nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot