human VPAC1 receptor is also validated for Aequorin (calcium), ERK1/2 and radioligand binding competition assays

Target Information

Family :
VIP-PACAP
Receptor :

VPAC1

Species :
Homo sapiens
Accession number :
NP_004615.2

Assay Information

Cat. Number :
FAST-0561C
Method :
HTRF
Assay Type :
cAMP – Gs mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
VIP
EC50:
9.1pM*
#ALT#

Mode:
antagonist
Reference antagonist:
PG 97-269
IC50:
291nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot